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BI-D1870 编号 : 122914

化学信息

产品英文名称BI-D1870
Iupac 化学名称2-(3,5-difluoro-4-hydroxyanilino)-5,7-dimethyl-8-(3-methylbutyl)-7H-pteridin-6-one 
同义词BI-D 1870 
英文同义词BI-D 1870 
分子式C19H23F2N5O2 
分子量391.415 
SmileCC1C(=O)N(C2=CN=C(N=C2N1CCC(C)C)NC3=CC(=C(C(=C3)F)O)F)C
InChiKeyDTEKTGDVSARYDS-UHFFFAOYSA-N
InChiInChI=1S/C19H23F2N5O2/c1-10(2)5-6-26-11(3)18(28)25(4)15-9-22-19(24-17(15)26)23-12-7-13(20)16(27)14(21)8-12/h7-11,27H,5-6H2,1-4H3,(H,22,23,24)
Cas501437-28-1

技术数据

外观Solid powder 
纯度98% 
可溶性Soluble in DMSO 
存储-20 ºC for 3 years 
运输条件Shipped under ambient temperature 
质量控制

产品详情

BI-D1870 is an ATP-competitive inhibitor of S6 ribosome for RSK1/2/3/4 with IC50 of 31 nM/24 nM/18 nM/15 nM, respectively; 10- to 100-fold selectivity for RSK than MST2, GSK-3, MARK3, CK1 and Aurora B. BI-D1870 also has a Kd value of 3.5 uM for BRD4. 

结构

122914 - BI-D1870 | CAS 501437-28-1

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