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EPZ011989 编号 : 120112

化学信息

产品英文名称EPZ011989
Iupac 化学名称N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-[ethyl-[4-[2-methoxyethyl(methyl)amino]cyclohexyl]amino]-2-methyl-5-(3-morpholin-4-ylprop-1-ynyl)benzamide 
同义词EPZ-011989; EPZ 011989 
英文同义词EPZ-011989; EPZ 011989 
分子式C35H51N5O4 
分子量605.82 
SmileO=C(NCC1=C(C)C=C(C)NC1=O)C2=CC(C#CCN3CCOCC3)=CC(N(CC)[[email protected]]4CC[[email protected]](N(CCOC)C)CC4)=C2C
InChiKeyXQFINGFCBFHOPE-WXUXXXNLSA-N
InChiInChI=1S/C35H51N5O4/c1-7-40(30-12-10-29(11-13-30)38(5)15-18-43-6)33-23-28(9-8-14-39-16-19-44-20-17-39)22-31(27(33)4)34(41)36-24-32-25(2)21-26(3)37-35(32)42/h21-23,29-30H,7,10-20,24H2,1-6H3,(H,36,41)(H,37,42)/t29-,30-
Cas1598383-40-4

技术数据

外观Solid powder 
纯度98% 
可溶性Soluble in DMSO 
存储-20 ºC for 3 years 
运输条件Shipped under ambient temperature 
质量控制

产品详情

EPZ011989 is a potent, selective orally bioavailable EZH2 inhibitor with Ki < 3 nM for EZH2 wt and EZH2 Y646; 15-fold selectivity over EZH1 and >3000-fold selectivity over other HMTase. 

结构

120112 - EPZ011989 | CAS 1598383-40-4

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